Cite tete wTapedetete anata ee Scheie catalan tne 7 - pas eee se rae ee i) i ‘iro ware we) heating trae TOXICITY OF 4,346 CHEMICALS TO LARVAL LAMPREYS AND FISHES SPECIAL SCIENTIFIC REPORT-PSHERES No. 207 UNITED STATES DEPARTMENT OF THE INTERIOR FISH AND WILDLIFE SERVICE EXPLANATORY NOTE The series embodies results of investigations, of restricted scope, intended to aid or direct manageme or utilization practices and as guides for administrativ or legislative action. it is issued in limited quantities official use of Federal, State or cooperating agencies processed form for economy and to avoid delay in publ United States Department of the Interior, Fred A. Seaton, Secretary Fish and Wildlife Service TOXICITY OF 4,346 CHEMICALS TO LARVAL LAMPREYS AND FISHES By Vernon C. Applegate, John H. Howell, A. E. Hall, Jr. Fishery Research Biologists Great Laxes Fishery Investigations U.S. Fish and Wildlife Service and Manning A. Smith Professor of Chemistry Bucknell University Special Scientific Report--Fisheries No. 207 Washington, D.C. March 1957 CONTENTS INTLOGUCEL ON Pejelelelelevete vole aleleielclelevelelelelcleleieieleiclcleleloleleleleleieieicleleieleleloleleieloleteielelstereletelo Preliminary screening Methods ..ceccccccccccuccccscccccsscccccccccccvccces Method of reporting screening test data .. ccccccccccvcccccccccccccccccccasece DISCUSSION .ecccccccccvescccceccccccescecceeccerececceseeceeceesescececee Acknowledgments ..ccccencccccccccccccccsccccsccccccccccccccccccccccccce WITELAtUTENCIUC cverc\ereleieie’elalevelelelelelovelele eleveleleielevele’elevelele(eleleleleleleleleleleleleteloieleteteroretele TABLES No. Bale Alphabetical list of 3,939 compounds with the results obtained in preliminary screening tests of each substance. scseseccccccccccccccce 2. List of 407 additional compounds, identified by code numbers only, with the results obtained in preliminary screening tests of ECACHESUDSTAN CE ores ele eisielsioielsleleleloieleleielelelelelelelcleleieleeicieleleyeleleleleleieleletelelelelsforets 3. Index of trade names of commercial products which are listed under systematic names in Table 1...ccccccccccccecccccscscocsccccce 4, Numerical list of sources of COMpOUNS. ececceccccccccccecscceccccccces De Alphabetical list of sources of compounds, ...cccccccccccccccccccccones bo 137 150 152 155 TOXICITY OF 4,346 CHEMICALS TO LARVAL LAMPREYS AND FISHES INTRODUCTION The problem of controlling the sea lamprey in the upper Great Lakes has received considerable attention in recent years and requires no review here (Applegate and Moffett, 1955), Electromechanical weirs and traps and electrical barriers have been developed which can be successfully employed to block and/or destroy spawning runs of adult sea lampreys. These devices, when installed in all known spawning steams, provide an effective method of reducing the numbers of sea lampreys in each lake basin. Initial efforts at control of the lamprey have employed these devices (Applegate, Smith, and Nielsen, 1952; Erkkila, Smith, and McLain, 1956). Unfortunately, however, a sea lamprey control program based on the prevention of spawning will not show results for seven or more years, At least six generations of larvae, spawned previous to the "blockade" of the streams, must grow, transform, migrate to the lakes, and prey on fish before the "blockade" is effective. Such a delay may prove disastrous in Lake Superior where there is evidence that lamprey predation will cause the collapse of the lake trout fishery, as has occurred in Lakes Huron and Michigan, before weir control measures can become effective. In view of these facts the principal problem is now one of developing techniques for attacking the sea lamprey which will produce more immediate control of the species, If we could destroy the larvae in the steams we might reduce substantially the parasitic populations in the lakes in less than two years, The introduction of natural enemies has been considered but invariably there is a great risk that “the cure might be worse than the disease", A more direct attack is provided by the use of either indiscriminate or selective poisons, Indiscriminate poisons, which would kill all fish-life in a steam, are undesirable since most streams infected with sea lamprey larvae also contain populations of important game and food fishes, The major objective of this investigation was, therefore, to locate chemicals which would be acutely toxic to larval sea lampreys at extremely low concentrations and which, at the same concentrations, would be non-toxic to other fishes inhabiting the same natural environments, The initial step in achieving this objective was a preliminary screening of a large and diverse seties of predominantly organic chemical substances. Test procedures in this program were designed only to disclose toxicity at low levels in short periods, The screening tests reyealed some compounds which, at particular concentrations, were more toxic to lamprey larvae than to fishes; others appeared toxic only to the larvae, Among these substances, only two were found to be sufficiently toxic and specific in their action at low concentrations to meet the tequirements and objectives of our program, Preliminary data for these two compounds and subsequent studies conducted to determine their usefulness as specific sea lamprey larvicides are not included here; they will be discussed in separate reports, The present report includes all other information obtained in the screening program on the apparent toxic effects of 4,346 compounds among larval lampreys and two species of fishes, These data are summarized here for the use that may be made of them by industrial chemists, toxicologists, physiologists, fishery scientists, and others, PRELIMINARY SCREENING METHODS All compounds were tested at an initial concentration of 5 p.p.m. Tests were conducted for a 24-hour period at a water temperature of 55 deg. F. Observations on the toxic effect of compounds were made on larvae of the sea lamprey (Petromyzon marinus) and also on rainbow trout (Salmo gairdnerii) and bluegill sunfish (Lepomis macrochi- tus). Larval lampreys varied from 3 to 5 inches in total length, Test fishes were of fingerling size, 4 inches or slightly less in length; every effort was made to keep size variation at a minimum, Larval lampreys were collected by means of an electric shocker in the Ocqueoc River, Presque Isle County, Michigan, and were held in running water in aquaria and small "races" under conditions which simulated their natural steam habitat, Test fishes were obtained from the stocks of local State and Federal fish hatcheries and were held in large raceways. These specimens were maintained in the best possible physical condition until used in the laboratory, Generally, two specimens of each of the three species were used in each test, Due to periodic difficulties in obtaining supplies of bluegills and rainbow trout, some compounds were tested using lamprey larvae and only one of these fishes; others were tested using only the larvae, The aggregate test animals available, usually six in number, were placed together in a 10-liter glass battery jar containing 5 liters of water, These jars were provided with aeration through standard stone air-breakers (at near oxygen saturation, as determined by repeated tests) and were maintained at a constant temperature by immersion in specially- constructed constant temperature troughs, These troughs were modified from a design described by Lagler (1953), Water temperature was maintained within the limits of $1.0 deg. F. Four such constant temperature units were utilized, each having a capacity of thirteen 10-liter battery jars (Figure1). Twelve of these test jars (each containing a substance being assayed) were included with one control jar in each trough, Fish and larvae in the control jar were exposed only to the water and physical conditions of the typical test container, Water used in all tests was drawn from a supply pumped directly from Hammond Bay of Lake Huron, The suction line intake of this pumping system was located 250 feet offshore at a depth of about 9 feet. Water from this source was consistently clear and of a relatively uniform quality, During a typical year while tests were being conducted (November 1953 to December 1954), pH varied from 7.5 to 8.2, dissolved oxygen from 8,6 to 13,7 p,p.m., and free COo from 5.0 to 9,0 p.p.m. Further data on the physical and chemical characteristics of northern Lake Huron water has been presented in a recent report by Ayers, Anderson, Chandler, and Lauff (1956). Chemicals were weighed in calibrated weighing bottles to the nearest milligram on a Volland Speedigram balance, Solubility of each compound was then determined in water, acetone, and ethyl alcohol (absolute), Five cubic centimeters of the indicated solvent was added to each sample, Each concentrated mixture was next added to a predetermined volume of water (as required by actual weight of sample and desired concentration) and agitated with a Power-Stir to produce a more dilute solution, Emulsions or suspensions of insoluble compounds were made with the aid of a Waring blender. These prepared solutions, emulsions, or suspensions were added to the test containers in which the experimental animals had already been placed, The resultant volume in each test jar varied from 5800 to 6200 ce. Knowledge of the degree of purity of many chemical samples was not available to us, All samples were therefore treated as "pure" preparations and the solutions at routine test concentrations were made accordingly. The specific content of some formulated materials was known while for others only incomplete data were available. For the sake of uniformity, all formulated compounds were tested at the routine concentrations used without regard for the proportion of active ingredient(s) present in each, The acetone or alcohol used frequently as a solvent exposed many test animals to concentra- tions as higii as 5 parts per 1000 of these substances. Repeated experiments were performed in which larvae, trout, and bluegills were exposed to the maximum concentration of each solvent that could occur in any screening test, No adverse effect on any species was observed at any time. Observations of each test were made approximately six times, at various intervals, during the 24-hour test period. At each observation, the condition of every test specimen was determined and tecorded, Chronological histories were thus obtained of any symptoms of illness and the occurrence of death, Any chemical killing the larval lampreys in eight hours or less at a concentration of 5,0 p. p.m. (regardless of the effects on other fishes) was tested further at levels of 1.0 and0.1 p.p.m. Water temper- ature, test period, and procedures were identical with those described for the initial test at 5.0 p. p.m. FIGURE 1, Constant temperature troughs utilized in the screening program, Concurrent tests of 48 different substances are shown in progress, Routine observations are being noted on the individual test record cards, Due to the large number of chemicals available for screening, it was not possible to test the majority of them in duplicate, nor was it considered necessary to do so to fulfill the objectives of the program, Where ambiguous results were observed, tests were repeated until definitive results were obtained, METHOD OF REPORTING SCREENING TEST DATA An alphabetical list of 3,939 compounds, with the results obtained in preliminary screening tests of each substance, is presented in Table 1, An additional 407 compounds, identified by code numbers only, are listed with similar test data in Table 2, Chemical nomenclature, as employed in Table 1, conforms to the Chemical Abstracts system, In many instances, related chemicals with entirely different names were received from different sources, For this reason, we felt it necessary to adhere to a uniform nomenclature system, The Chemical Abstracts system was adopted because its basis is readily available [See: Subject Index; “Introduction, with key and discussion of the naming of chemical compounds for indexing", Chemical Abstracts, Vol. 59 (1945), pp. 5867-5975]. In most cases, consultation of the Fourth Decennial Index or the annual index of a recent year of Chemical Abstracts will suggest the manner in which we have listed a particular class of compounds, Inverted names have been used for substituted compounds, The inverted portion either follows a comma after the parent name or receives a first order of indentation, The substituents are in alphabetical order, Other modifications of the compounds (salts, esters, commercial formulations, etc.) are either separated from the name by a semicolon or receive a second order of indentation, In a few cases, a rational formula could not be constructed from the name given by the supplier, When attempts to resolve this difficulty failed, the name has been entered in the table as received, Materials of unknown or doubtful composition are listed by the name provided by the supplier, In some instances, trivial chemical names have inadvertently found their way into our list (nearly all of these are cross-referenced in the Chemical Abstracts subject indices). A number of commercial chemical products were tested in the screening program, Where the chemical identity of these substances was not immediately available, they have been listed directly in Table 1 by trade name. Other products, whose identity was known to us, have been given primary listing by their proper chemical names, A cross-reference index is presented in Table 3 which will aid in locating the latter group of commercial compounds in Table 1, For simplicity of tabular presentation, any toxic effects of compounds have been expressed in terms of the elapsed time of exposure required to produce some obvious pathological condition, Thus, the figures given in Tables 1 and 2 indicate the time in hours, fractions of hours, or minutes to cause death or obvious distress. Each time datum represents the average response of all test specimens of a particular species, Private concerns, public agencies, and individuals that supplied the compounds tested have each been assigned an identifying number, For tabular convenience, these numerical designations have been utilized in Tables 1 and 2, They may be identified by reference to Table 4 which is a numerical list of sources, An alphabetical list of these sources with their identifying numbers will be found in Table 5, DISCUSSION The screening test data presented in this report should be viewed only as indicative of the toxicity of the individual compounds, Our objective was limited to the identification of biologically active agents that would be selectively lethal to larval lampreys. Laboratory procedures did not permit the numerous test replications necessary for positive definition of the toxicity of each substance, For this reason, conventional toxicity ratings have not been computed, Test results obtained with many compounds were undoubtedly influenced by the quality of the water used, It should be borne in mind that widely divergent results with any particular compound might be obtained were these tests to be repeated in waters possessing different chemical and physical properties, Repetition of test: utilizing hatchery strains of fishes, other than those employed by us, might also produce some variation in results, Many similar substances were present in the large series of compounds which we tested, The aggregate data available for some groups of related chemical structures is considerable. These collective data may provide clues or suggestions to investigators who are interested in the nature of any biological activity which characterizes the members of a related group of substances, Of particular interest is the rather marked specificity seemingly displayed by certain compounds, Among those tests where all three species were exposed, 264 of the substances were toxic to only one species at the levels of concentration and temperature employed (included in the preceding total are the two substances, omitted from this report, which merited extensive investigation as possible sea lamprey larvicides). Three hundred and thirty-three additional compounds were toxic to only two species while displaying no evident adverse effect upon the third, These observations are derived from the data recorded in Tables 1 and 2; no separate listing of these particular compounds has been prepared, The nature of our objectives has permitted us to do little more than note the aforementioned evidences of specificity, Critical studies are required to evaluate the precise biological activity of each of these substances, Many of them may prove to be of little practical value in the light of such studies; others may demonstrate a useful selectivity that can find application in fish population control techniques. It is hoped that the necessary further research suggested by our findings will be undertaken, ACKNOWLEDGMENTS Nearly all of the chemical samples tested by us were originally assembled for use in another investigation by the staff of the USFWS Microbiological Laboratory at Leetown, West Virginia, Shortly after the conclusion of their study, these samples were made available for our screening program, We are indebted to Dr. S. F, Snieszko, Director of the Microbiological Laboratory, and to Dr, Robert E, Lennon and Philip S, Parker for their cooperation and assistance in the transfer of sample materials, records, and related correspondence, We are also grateful for their advice and suggestions concerning screening program techniques, The investigations conducted in both laboratories would have been impossible without the outstanding cooperation displayed by the many private concerns, agencies, and persons who submitted compounds for testing. In the further use which we made of their samples in our study, we frequently required additional chemical data or supplemental supplies of many compounds, These were kindly provided by the contributors wherever it was possible for them to do so, We particularly appreciate their generosity in permitting the chemical identification of most of their materials in this report. All rainbow trout and most of the bluegill sunfish fingerlings used in our tests were provided by the Fish Division of the Michigan Conservation Department, Over 40,000 of these fishes were delivered by the Department to our laboratory in small, periodic consignments, Mr. M. J. DeBoer, Supervisor of Hatchery Operations for the Fish Division, was largely responsible for coordinating delivery of the fish, His assistance, and that of other hatchery personnel of the Department, is gratefully acknowledged, In addition to these specimens, one consignment of bluegill sunfish fingerlings was received by us from the Rochester (Indiana) Fish Cultural Station of the Fish and Wildlife Service. Dr. James W. Moffett, Chief of the Service's Great Lakes Fishery Investigations, participated in the planning of the investigation and contributed much administrative assistance which expedited our work, Mr, John F, LesVeaux of the Research Department of the Niagara Chemical Division, Food Machinery and Chemical Corporation, provided valuable technical advice, consolation, and suggestions concerning methods of reporting our data, During the extended period the screening program was underway, numerous technical and clerical assistants joined our staff for varying periods of time. Among those who demonstrated exceptional interest and initiative in their duties were; Clifford L, Brynildson, Clyde O, Barr, Chester J, Pszczolkowski, Rose L. Hoffman, Norma J, DeMara, Mary E, Dimick, Clarence H, Barrette, Clifford R, Kortman, and Margaret A, Evans, The manuscript and tables for this report were typewritten for direct reproduction by Martha A, Bergen, Many other persons, not associated with our staff, contributed advice and assistance which were of material aid in the investigation, LITERATURE CITED Applegate, Vernon C, and James W. Moffett 1955, The sea lamprey, Scientific American, Vol. 192, No. 4 (April), pp. 36-41. Applegate, Vernon C,, Bernard R, Smith, and Willis L. Nielsen 1952, Use of electricity in the control of sea lampreys: Electromechanical weirs and traps and electrical barriers, U. S., Dept. of the Int., Fish and Wildl. Serv. , Spec, Sci, Rept.: Fisheries No, 92, 52 pp. Ayers, J. C., D, V. Anderson, D, C, Chandler, and G, H, Lauff 1956, Currents and water masses of Lake Huron, Great Lakes Research Inst, (Michigan), Tech, Paper No, 1, 101 pp. Erkkila, Leo F,, Bernard R, Smith, and Alberton L, McLain 1956. Sea lamprey control on the Great Lakes - 1953 and 1954 U. S. Dept. of the Int,, Fish and Wildl, Serv., Spec. Sci. Rept: Fisheries No. 175, 27 pp. Lagler, Karl F, 1953, Constant temperature bath for experimental aquaria in linear series, Copeia, 1953, No. 4, p. 242, TABLE 1, Alphabetical list of 3,939 compounds with the results obtained in preliminary screening tests of each substance. EXPLANATION OF TABLE Chemical nomenclature follows generally the Chemical Abstracts system; certain exceptions are noted in the text, Sources of compounds as indicated in the columns headed "Subm, " may be identified in Table 4, Submitters code numbers are those used by the suppliers to identify their own materials; those known to us are listed herein, Tests at indicated concentrations were conducted for a 24-hour period at a water temperature of 55 deg. F, Formulated materials were tested at the routine concentrations used without regard for the proportion of active ingredient(s) present in each, Figures given indicate time in hours, fractions of hours, or minutes ("m,") to produce death or obvious distress and are the average response for each species (where illness only was observed during the test period, the average time to produce this response is underlined); an "n" indicates that no effect of the chemical was observed; a dash indicates that the test was not performed; the names trout, bluegill, and lamprey larvae are abbreviated T, B, and SL respectively. - =! % - See ac) care nal - (TAtTeTAtpout-Z) -N-010749-,Z TSL=9 ig 88 - - - - - - Lie Co - (Axomaoro[yp -Z) -,Z 068-10 hig 98 & = = = - - me -010[ 49-7 Z1e-ID fe C =, - - = 5 u u u -O1O[Y9 =Z €TE-ID LS TE ja = = 2 = Z u u u -O10[ =D 08% ‘006 SZC - 2» ee Or u FL OF -kxospky-Z -1Aang-1101=¢ 669-ID LG) = - - - - - u u u -1Atpe (Axomatxoing-Z) -Z-N IZ0T-I0 i E G = 3 = 2 ie nu Skt -ouloiq=¢ 860 ‘S06 fife = S = = = = u u u -Kxojkzuoq-,Z ZEP-IO Ig= 9% - - - - = ~ u = = -ouyure=d ZZ 9% 8 - - - - - - Uru u -[Ainq-1101-g-A£x01008 -Z 869-10 Ka 5% = = Ss o - - u u u -ontu-d-0100"-pD ‘apTtiueis0y 90€-ID LS 8% = = = = = = u u u Joiso [Amoor0TYyO-g !-or0T Yorn T-WS LS ZS - - = - - - ie) ee) -tAtretktpout-g-N]] stq (eusyueyd=d) -,N ‘N 6FL=ID i = Vie ~ = = = = S u u u -TAtretAneut-g -N] stq (auatAusyd-t) -,N ‘N 06-10 LG 0Z S = = ‘= co = u ae u - ({Ataydeu-g-ontu-T) -N 63-19 ES 6 - - - - - - Ge th - ((Awpydeu-Z) -N 983-ID LS L¥0 TOS eZ 8 s = " 2 - = it) tite at - (tAmpydeu-T) -N 8r0 ‘TOS a hi - - - - - - i Sat - (tAuydeu-T) -N- (tAtretAtout~Z) -N. 6EL-ID hy OV haa = = om = c= FI v vA -[Azettpozueg-g-n -oideosoul-p 9LT-OT LS CL - - - - - - Oh = Se hn - (xotpekxomphy-Z) -Z ges ‘OTS fh a 2 3 s = 2 = u u u -[Auaydtp-N *N. 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B6BE ‘ = . = 7 _ u u u apAyapleneiaA IST 9F ~—s T68E a = . = = 2 u u u qoi1so [Aupa ‘pyoe OTTTUEA PI 9 ~—- 068E - - - - - - u - - -TpAxo-,¢‘g ‘atIntuoieyeA = TE. “00S GS 6886 5 E = ~ = - u - z aTIMMoo[ZoueINj-Z YIM Jolso !-onyu-p-[Aoul-7 L@T-Ua LS 8888 - - - - - - u - - qaiso [Ato !-oul0%q-¢ ET ‘E0P GZ L888 - = = - - - u - - wes (11) [eyoTU ‘proe oreyeA = 8 9- 98h “LOT GZ 9888 = = = Es S < u - = proe on = 90 *T0S GS G88E 1S qd it AS At, Sued AT “ON T°0 Ona ons 2pod pon uidd ut uonenusou0D [eOTUISYD Jo ouIeN *uiqng ‘uiqns ‘I1doy 134 SFARAOA AG aa SSeS Oe ie ees ee OY ISO tsb ss) PME aies Tai {=} a 4 S Oo aan i SN ents EP SOE TAIIEE eyteh Ih te on =) VT ~OIONTJEXOY =, *o ve ‘ 9 ‘6 apHoryoorpAy touapr{{x-¢ °Z -tAqrerdtout-g-N ‘outpiyAx-x *x joust{x =< *¢ -or0Tyo= (4) (9 pue)zg jous|kx-F *¢ jousth{X-F *Z proe oruos;nsoustkxed Tes WMIpos ptoe oTuoj~nsausyk{x-o ayes umMTpos plor oTuoy;nsaue,AX-ur Joiso [Auoyd qaisa [Aoapop saisa [A{kuaydiq-7 ‘prior oTuojy[nsouatAK~-x -[AtmooueAoTp-N *N Saprureuoypnsauapkxed -oTu -o10[yorp-,p *v ‘auethx-d -o1oppexoy~9 *c *P*e *,D*p -o10[YoIp-,p ‘pv *auatkx-0 - [Axomme (Axomakxoyhzuoq-2) -g] -p-AxopAzuaqip-,p *p - (Axomokxophzueq =z) -p-Axophzuoqip-,p *p *auayXx-ur jorpAyue x auomue x DAMPATIOp uMTpos ‘*Joiso [AIPoTp ‘pfoe OTuOpTreyootpue xX rojso [Auiogosy {prow oMeovotpuRNX apytnsompAyue oppure x aptuieoodT3 AIM Jalsa !~[A1uod rajso [Apa !-[Auoydosoyypeiuad aieuoqmeopormpyAIe-O IIM opTyTNsospAyur ‘-;Atpo ‘pror ofmueKX ¥CS *008 STS 6ZL-ID 133 “80F 6S “O0T LS *O0T ZESS-O d- 0613-O TeZS-O d- L61Z-O Z2S-O ZP9Z-O FSLZ-O 6F9Z-O 60LE-O 888 T-dN 680 ‘000 LLP-2H 6LP-9H 88T 68 S9- 819 ‘90T SSEP-O OT-07T 961-01 L¥0 “TOP 9P GG LE6E 9E6E SE6E VE6E €6E 86E TE6E Of6E 6368 826E LZ6E 9268 S36E Vo6E €36E 326E T36E 0268 6T6E 8T6E LT6E 9T6E ST6E PI6E S168 ST6E TT68 OT6E 6068 8068 135 a LMM mac. —. ..°: _ . o uT uoMeQUeDUOD TeOTUIaYD jo ouleN OPHONTJOOIIs OUTZ 59D qresiyoouodez 890 °004 apoD *ulqns 9 SZ *ulqns °ON doy 136 TABLE 2, List of 407 additional compounds, identified by code numbers only, with the results obtained in preliminary screening tests of each substance, EXPLANATION OF TABLE Names of these compounds have been restricted by their submitters, Compounds have been grouped by source and, for each submitter, are arranged alphabetically and/or numerically according to the submitter's own code numbers, In all other respects the presentation of data here is identical with that to be found in Table 1 (See Table 1, “Explanation of table", page 9). 137 u u u gu u vv Ab 8 9099-S 9S 9968 < _ Ss = = = 6 6 I 16Z9-S 9S G96E fe & = = = x u = = CPI-S 9 P96E - 5s & Z - = Aa ea 8PPI-dN 9g 6968 z = 2 3 “i E i LUVI-dN 9g 2968 = = S = = = u u u ZLVI-dN 9¢ T96E < = 5 = - - Bib 42-16 VOET-dN 9¢ 0968 = = Z : “ = at. tt 6 ES8T-dN 9S 6S68 u Tiere u u u Ds g G831-dN 9g 8S68 - = = - - - Clee T VOZI-dN 9S LS6E = £ = é = - u eo SSTI-dN 9S 9968 u ue wu ae AG z g I I €80T-dN 9S sc6s a = = = = a U u u 8POT IZP-WNS LS 9LTP 3 3 x e 2 z u = = 0ZF-NS LS SLIP 2 “ 2 é < 3 Teens - 9TP-NS LS PLIV 2 a 2 2 2 “ uae 2 2 IIP-NS LS SLIP = s - = “ 2 mi -2 = LOv-WS LS ZLIv z é 3 s : Z u 3 = 8t6-NS LS ILI 2 2 2 i 2 s u g . 908-INS LS OLT s 2 3 2 = = W = fh BR T6Z-WS LS 69TP = “ - z “ z Tee ime ee! 482-0 LS 891 = 5 9-8 - - - Bie 283-0 LS LOI = < z 2 “ Ties eet 18Z-0 LS 99TPr Z “ 2 x a 2 ie 2 = CLZ-O LS Solr “ is e 2 s = we <6 2 692-0 LS VOIP z 2 = = = = Ue ue 162-0 LS eolr s « = 3 3 = u u u 6%Z-O LS ZOTV = E = Z < 2 i oe an 022-0 LS I9TP S < z 3 Fs = u u u TIZ-O LS O9TF S = = 6 O = u u u L6T-O LS 6STP 2 3 2 z “ - Ge = oe VET-O LS 8STP é = E : 2 © Wes 2 LZI-O LS LSTP - 3 s 2 E 2 ae ZBI-O LS 9STP 2 a « 2 a 3 ie 2 a 8102-0 LS Sct = 5 2 = = z ee cue 010Z-O LS VSP = 2 : s = 2 u . = €0LT-O LS esly F 2 2 z 2 = i une ZOLT-O LS 2SPr z - - = - - en yee CT 09-31N LS IST = = os 2 © = u u u 9¢-IIN LS OST? Ts qo 2 Rin Gln aa See ae: "ON Tn Oat 0's apoD “ON uidd ut uonenuesuo5 *uIqns *ulqns doy 144 wot dan ESO nmanrnraAaNARRFANAARAERE AMA eE AA eee eaaaat asa aeamaeaso wt T8-A TL-A c9-A €9-A cc-A 8h-A Lb-A vE-A Té-A 66-A 86-A €Z-A 03-A 6T-A 8T-A LT-A €T-A TT-A OT-A v-A T-A S6S-WS LLS-WS TLS-WS OLS-WS G9S-INS POS-INS €PG-WS GéG-INS VES-WS €es-WSs 82S-INS 96S-WNS T3S-WS 03S-INS 80S-INS 96P-INS 06P-NS 68P-INS E667 66SV 1630 0337 6167 8IZV LIGV 9T3V ST3V VIP €1SP SlsP TT3P OT3P 6067 8067 LO&P 906P S03P VOSP £037 B0ZP T03P 006% 661P 86TP L6OTY 96 TF S6IP VOTP S61P 66TP T6TP O6 TP 68TP 88TP L8TV 98TY C8tP 145 a — o C = = u u u €6Z-A LS 8S67 & Bs 2 c = = u u u Z6G-A Lg LSZV Bs 2 = = 2 = u u u 06Z-A LS 9827 7 2 = bs 2 z U u u 88-A LS GGar = 2 é = = 2 u u u 6LZ-A LS HOSP u u u u 6 u Re GE g 89S-A LS ES37 e a = = = - we G9 6SZ-A LS ZSBP S z 2 2 2 3 u €l ou LSZ-A LS TSZP 5 = es - = - We Gat GSZ-A LS 0S3r 2 2 x é 3 S u u u LVB-A LS 6VEP = = = = = : u u u FES-A LS 8hCP 2 = = = Ss . G1 u S8T-A LG LVGY 3 = = 2 = = u u u €8T-A LG 96D : < = = - - 6 g z LLT=A LS SvEP 5 = E = = = u u u GLT=A LS aA = = - - - - tL 9 v 89T-A LG EPBP u u u ¥ tL 6? a7 & T LOT-A LS SOP s = = 2 = = u u u 99T-A LS MA = = = = - - u u &I ZOT-A LS OVEF - 2 2 5 5 = u u ¥ T9T-A LS 6EZF E 3 2 x = £ u 2 = OPT-A LG 8ESP = = z 2 s z u u u ZET-A LS LEG - = = 2 = = u u u O8T-A LS 9ESP = : = 3 = = u u u L3T-A LS SEZr a - Z = : x u WL Ou 9ZT-A LS ECP = = = = z z u u u STI-A LS 8ESP - - = - - - Ve 4k. te PLI-A LS ZESP = = = a = = u u u TLIT-A LS TESD = = a = = = Ci ac g OTT<-A Lg era - = = = = = u u u LOT-A LG 6337 3 4 = = = = u u u G0T-A LS 823P z = = = S = u u u TOT-A LS LSP Z a = ~ = = u 2 = C6-A LS 9BBF = = = = o = u u u Z6-A LS SZSV = = = = = = u 5 = T6-A LS aca 1S d ‘it Ser af, ASH L *ON 130 OE 0°S 2pod gON ul uONe DUaDU0D *uqns *uqns "doy 146 a u =] a ae (a wm aw ws N bo ho | APA RAR Ae aor er ae aana aH al eo nc ateaa WANE BMDNANANHINGUAN AON AG PH a BemwttaeanWtnAAReARaNnNnaeas Neen GC GNanwn ni NN aN GAA 4 =e Naomi CWORRN KR RAN Ret cw -_ LS LS LS LG LS LS LS LS AS LS LS LS LS LS LS LS LS LS LS LS LS LS LS LS LS LS LS LG LS LG LS LS LS LS LS LS LS LS 9660 S630 VEST 667 6630 T6367 0667 6867 8867 L860 9867 S86P P8Er E837 S86P T837 0867 6L3P SLOP LL&P OLED GLEY PLOY SLOP SLOV TLV OLZP 69h 893P LOBE 996P S9GP PISP 696P B96P T9360 0987 6S6P 147 = 2 = = - = u - - L-TT8¥-O 69 TZ8V = é : ~ = 3 u - - 9-TTEF-O 69 0ZEF : = s = = z u - - G-TIEF-O 69 6187 = S z co a S u - - €-LI8h-O 69 8&7 = z = = = = u - - Z-LI€F-O 69 LI&? s 5 2 © 2 = u - - T-LI€F-O 69 9TEV z = = = S = u - - 908%-O 69 GTer z < 5 = S = u - - S08h-O €9 vIEP = = : = 2 = u - - $9Z7-O €9 eter = = a = z = u - - 6S37-O 69 ZleP 2 e = o ~ 5 u - - TIZP-O 69 TIep = = = = = = u - - 8067-0 €9 OTEY = S = = = - u u u 3STP-O £9 6087 = = = = = = u - - L90%-O €9 807 = = = 6 = = u - - Z16E-O 69 LO&? = = - C = = u - - V¥8Z-O 69 9087 = é = = - = u - - 8682-0 69 SOET 5 . = a = = u = - 9D-0%LZ-O €9 POST = zs : a = = u u u d-0LSZ-O 69 €0EF = = & = a = FI ou u @G-dd (ay) S0EV s = = S & = u - - 909F-dD 6S TOEr - = = - - - u u u S886 -dD 6S 008% = _ 3 = = z u - - 688-dD 6S 66h = = “ a = & u u u 8E8-dD 6S 8627 = S = < = = u u u 8Z8=-dD 6¢ L667 1S Gi ie 1s 4 At AS een *ON Lo@ 0°T 0°S 2Ppod ON uidd ut uopequosu0D *uqns *uuqns doy 148 1 1 i i fh Tepes) tobe(s eth (=) Ta) a fet ep tey ael at fel ist teh is) 1 i i] 1 a = 1 1 1 i 5 O-38SS-O H-Z8SS-O 9-G8SS-O 09SS-O €87S-O S86S-O I-LSES-O 6VES-O OTES-O L83S~-O 3S3S-O 60TS-O III-8SL¥-O II-8SL¥-O S09P-O 98SP-O T6bp-O d-8L¥V-O d-S9PP-O V-S9bP-O TL0ry-O 8687-0 L8EV-O BPEV-O vEEP-O €9 €9 €9 €9 €9 €9 €9 €9 €9 €9 €9 €9 €9 €9 £9 €9 €9 €9 £9 69 £9 €9 £9 £9 €9 9VET SVED DEP Cver CVET Ter OEP 68EV Seer LEEP 98EP Seer PEEP Seer seeV TSP OfeP 668 828P LOEP IEP SEV POEV sev Bo8VP 149 TABLE 3, Index of trade names of commercial products which are listed under systematic names in Table 1, Trade name Subm. Rept. No(s). Actamer (59) 2876 AD-IT (34) 2465 Alanap-1 (55) 2989 Alanap-3 (55) 2990 Ammonyx DME (18) 287 Armeen C (11) 1194 Armeen 8 (11) 2572 Armeen 10 (11) 1361 Armeen 12 (11) 1454 Arneel C (11) 1195 Arneel 8D (11) 2546 Arneel 10 (11) 1348 Aroclor 1242 (58) 858 Aroclor 1248 (58) 859 Aroclor 1254 (58) 860 Aroclor 1260 (58) 861 Arquad 12 (11) 290 Arquad 16 (11) 291 Blueberry Dust (50) 987, 1201 BTC (18) 267 BTC-471 (18) 270 BTC-824 (18) 266 BTC-927 (18) 269 Chipman 6# Livestock Spray (33) 3792 Chipman 20% Dust (33) 3793 Chipman 40% Spray Powder (33) 3794 Chlordane (28) 1457 (See also: Rept. Nos, 1170-73) DDT (46) 1570 Dichlorobisphenol A (54) 866 Dilan (42) 2632 DN Dry Mix No.1 (28) 2785 DN Dry Mix No, 2 (28) 1227 Dow Defoliant (28) 66 Dow General Weed Killer (28) 2747 Dowicide A (28) 2868 Dowicide G (28) 2863 Dowicide 2 (28) 2878 Dowicide 2S (28) 2879 Dowicide 6 (28) 2871 Dowicide 31 (28) 2782 Duomeen C (11) 8103 Duomeen 12 (11) 3107 150 TABLE 3, (Continued) Trade names Subm, Rept. No(s). Emulsept (51) 3283 Fish= Tox (3) 3419 Isothan DL-1 (18) 286 Isothan Q-15 (18) 2127 Lindane (25, 36, 39, 42) 1264 to 1266 Naphthenic acid D (8) 2462 Noxfish (2) 3418 Nuodex Mercury (34) 2464 Nuodex PMO 10 (34) 2597 Onyxide (18) 288 Phygon Technical (55) 2491 Phygon-XL (55) 2490 Pluronic F-68 (63) 2593, 2594 (See also; Rept. No, 3051) PMAS (24) 143 Polyrad 1100 salt (1) 114 Polyrad 2000 salt qd) 115 Ryanicide 100 (2) 3421 Sindar G-i1 (19) 1515 Sorbit AC (14) 2454 Sorbit P (14) 2455 Spergon (55) 167 SUPER AD-IT (34) 3506 Systox (23) 2981 Tarophen CNB 33 (28) 499 Tetrosan (18) 268 Tolane (58) 211 Vancide 51 (38) 7112 Vancide 76 (38) 1022 Weedex (16) 3459 151 (1) (2) (3) (4) (6) (7) (8) (9) (11) (12) TABLE 4, Numerical list of sources of compounds, [Private companies, public agencies, and individuals who supplied the compounds used in screening tests are listed in order by the identifying number assigned to each. These identifying numbers are utilized in Tables 1 and 2 in the columns headed "Subm, "]. Naval Siores Department Hercules Powder Company Wilmington 99, Delaware Research Division S. B, Penick & Company 999 West Side Avenue Jersey City 6, New Jersey Vis-Ko, Incorporated Sumner, Washington Research Laboratory Geigy Agricultural Chemicals Geigy Chemical Corporation 62 West Second Street Bayonne, New Jersey Technical Service Department Davison Chemical Company Baltimore 3, Maryland Product Development Department Solvay Process Division Allied Chemical & Dye Corporation 61 Broadway New York 6, New York Oronite Chemical Company 3508 Carew Tower Cincinnati 2, Ohio Research Department Ozark-Mahoning Company Tulsa 1, Oklahoma The Market Development Department Armour Chemical Division Armour and Company 1355 West 31st Street Chicago 9, Llinois General Sales Offices Sumner Chemical Company, Inc, 6 East 45th Street New York 17, New York 152 (14) (15) (16) (17) (18) (19) (21) (23) (24) (25) Geigy Industrial Chemicals Geigy Chemical Corporation 89 Barclay Street New York 8, New York Government Contracts and Sales Mallinckrodt Chemical Works Second and Mallinckrodt Streets St. Louis 7, Missouri James Good Company Susquehanna Avenue & Martha Street Philadelphia 25, Pennsylvania Technical Service Department Chas, Pfizer and Company, Inc, 630 Flushing Avenue Brooklyn 6, New York Research and Development Laboratories Onyx Oil and Chemical Company Warren and Morris Streets Jersey City 2, New Jersey Sindar Corporation 330 West 42nd Street New York 36, New York Coahoma Chemical Company, Inc. P. O. Box 728 Clarksdale, Mississippi Chemagro Corporation 101 Park Avenue New York 17, New York W. A. Cleary Corporation New Brunswick, New Jersey The Chemical-Biological Coordination Center National Research Council 2101 Constitution Avenue Washington 25, D. C. (28) (27) (28) (30) (31) (32) (33) (4) (35) (3%) (38) TABLE 4, Sharples Chemicals Division Pennsylvania Salt Manufacturing Company Three Penn Center Plaza Philadelphia 2, Pennsylvania Battelle Memorial Institute 005 King Avenue Columbus 1, Ohio Biochemical Research Department The Dow Chemical Company Midland, Michigan (Restricted) Agricultural Research Division Shell Development Company P, O, Box 1531 Modesto, California Heyden Chemical Corporation Garfield, New Jersey Cincinnati Division Toms River - Cincinnati Chemical Corporation Evanston Station Cincinnati, Ohio Research Division Chipman Chemical Company, Inc, Bound Brook, New Jersey Microbiological Laboratory Nuodex Products Company, Inc. Elizabeth, New Jersey Product Development Department Shell Devélopment Company Emeryville, California Ethyl Corporation 100 Park Ave, Bldg, at 41st Street New York 17, New York R. T. Vanderbilt Company 230 Park Avenue New York 17, New York (Continued) (39) (40) (42) (43) (44) (45) (46) (47) (48) 153 Research Department Commercial Solvents Corporation Terre Haute, Indiana Southern Chemical Division The Glidden Company P. O. Box 389 Jacksonville 1, Florida Field Laboratory California Spray-Chemical Corporation P. O. Box 120 Haddonfield, New Jersey Niagara Chemical Division Food Machinery & Chemical Corporation Middleport, New York Agricultural Research Division Shell Development Company P, O. Box 2171 Denver 1, Colorado Naval Stores Research Section Southern Utilization Research Branch Agricultural Research Service U. S. Dept. of Agriculture Naval Stores Station Olustee, Florida Dr. W. T. Sumerford Director, Pharmaceutical Chemistry Research Laboratories Mead Johnson and Co, Evansville, 21, Indiana Process Research Department Chemical Division Merck and Company, Inc. Rahway, New Jersey Chemical Control Department The American Agricultural Chemical Company 50 Church Street New York 7, New York (49) (50) (51) (52) (53) (54) (55) (56) (57) (58) TABLE 4, Research Department Ringwood Chemical Corporation Woodstock, Llinois Department of Entomology University of Maine Orono, Maine Emulsol Chemical Corporation 59 East Madison Street Chicago 3, Illinois Hydraulic and Sanitary Laboratory College of Engineering University of Wisconsin Madison, Wisconsin Department of Botany and Plant Pathology Colorado Agricultural and Mechanical College Fort Collins, Colorado Research Laboratory Columbia~-Southern Chemical Corporation Barberton, Ohio Agricultural Chemicals Development Naugatuck Chemical Bethany 15, Connecticut Technical Division Pennsylvania Salt Manufacturing Company Box 4388 Philadelphia 18, Pennsylvania Research Laboratories Rohm and Haas Company 5000 Richmond Street Philadelphia 37, Pennsylvania Entomology Research Branch Agricultural Research Service United States Department of Agriculture P, O. Box 3391 Orlando, Florida 154 (Continued) (59) (60) (62) (63) (64) (65) (66) (67) (68) (69) Development Department Organic Chemicals Division Monsanto Chemical Company 800 North 12th Boulevard St, Louis 1, Missouri Velsicol Chemical Corporation 330 East Grand Avenue Chicago 11, Illinois Doe Run Plant Olin Mathieson Chemical Corporation P, O, Box 547 Brandenburg, Kentucky Research and Engineering Division Wyandotte Chemicals Corporation Wyandotte, Michigan New Product Development Department American Cyanamid Company 30 Rockefeller Plaza New York 20, New York Agricultural Chemicals Research Laboratory General Chemical Division Allied Chemical & Dye Corporation P, O. Box 405 Morristown, New Jersey Research Division Dr. Salsbury 's Laboratories Charles City, Iowa Division of Industrial Chemistry Commonwealth Scientific and Industrial Research Organization Box 4331, G.P.O., Melbourne, Victoria, Australia Eastman Organic Chemicals Department Distillation Products Industries Rochester 3, New York Biochemicals - Development B, F. Goodrich Chemical Company Rose Bldg. 2060 East Ninth Street Cleveland 15, Ohio TABLE 5, Alphabetical list of sources of compounds, Submitters name Submitter 's number Allied Chemical and Dye Corporation, General Chemical Division (65) Solvay Process Division (7) American Agricultural Chemical Company, The (48) American Cyanamid Company (64) Armour and Company, Armour Chemical Division (11) Battelle Memorial Institute (27) California Spray-Chemical Corporation (42) Chemagro Corporation (23) Chemical-Biological Coordination Center, The (25) Chipman Chemical Company, Inc, (33) W. A. Cleary Corporation (24) Coahoma Chemical Company, Inc. (21) Colorado Agricultural and Mechanical College, Department of Botany and Plant Pathology (53) Columbia-Southern Chemical Corporation (54) Commercial Solvents Corporation (39) Commonwealth Scientific and Industrial Research Organization, Division of Industrial Chemistry (67) Davison Chemical Company (6) Distillation Products Industries (68) Dow Chemical Company, The (28) Emulsol Chemical Corporation (51) Ethyl Corporation (36) Food Machinery and Chemical Corporation, Niagara Chemical Division (43) 155 TABLE 5. Submitter's name Geigy Chemical Corporation, Geigy Agricultural Chemicals Geigy Industrial Chemicals Glidden Company, The, Southern Chemical Division B. F. Goodrich Chemical Company Hercules Powder Company Heyden Chemical Company James Good Company Mallinckrodt Chemical Works Merck and Company, Chemical Division Monsanto Chemical Company, Organic Chemicals Division National Research Council Naugatuck Chemical Nuodex Products Company, Inc, Olin Mathieson Chemical Corporation Onyx Oil and Chemical Company Oronite Chemical Company Ozark-Mahoning Company S. B, Penick and Company (Continued) Pennsylvania Salt Manufacturing Company, Sharples Chemicals Division Technical Division Chas, Pfizer and Company, Inc. Ringwood Chemical Corporation Rohm and Haas Company 156 Submitter's number (4) (14) (40) (69) (1) (31) (16) (15) (47) (59) (25) (55) (34) (62) (18) (8) (9) (2) (26) (56) (17) (49) (57) TABLE 5. (Continued) Submitter's name Dr, Salsbury‘s Laboratories Shell Development Company, Agricultural Research Division (Modesto, Cal.) Agricultural Research Division (Denver, Colo.) Product Development Department Sindar Corporation Sumerford, Dr. W. T. Sumner Chemical Company, Inc. Toms River = Cincinnati Chemical Corporation United States Department of Agriculture, Agricultural Research Service, Entomology Research Branch Southern Utilization Research Branch University of Maine, Department of Entomology University of Wisconsin, Hydraulic and Sanitary Laboratory R. T. Vanderbilt Company Velsicol Chemical Corporation Vis-Ko, Incorporated Wyandotte Chemicals Corporation, Research and Engineering Division 157 Submitter's number (66) (30) (44) (35) (19) (46) (12) (32) (58) (45) (50) (52) (38) (60) (3) (63) INT.-DUP. SEC., WASH., D.C12798